SMALL MOLECULES
Insulin secretagogues |
Sulfonylureas, meglitinides, glucokinase activators, GPR40, GPR119, GPR44 agonists |
Insulin sensitizers |
Biguanides, PPAR agonists, SARMs, SIRT1 activators, 11beta-HSD1 inhibitors |
Incretin/glucagon pathway modulators |
Dipeptidyl peptidase-4 inhibitors, glucagon-receptor antagonists |
SGLT-2 Inhibitors |
Other oral agents |
Diacylglycerol acyltransferase and ACC inhibitors, thyroid hormone receptor beta (TRβ) agonists, farnesoid X receptor (FXR) agonists, peroxisome proliferator-activated receptor, niacin derivatives, CCR2 antagonists, ileal bile acid transport (IBAT) inhibitors, PDF4 inhibitors, de novo lipogenesis (DGAT, SCD1 & ACC) inhibitors, cannabinoid 1 receptor modulator |