SMALL MOLECULES

SMALL MOLECULES

Insulin secretagogues
Sulfonylureas, meglitinides, glucokinase activators, GPR40, GPR119, GPR44 agonists
Insulin sensitizers 
Biguanides, PPAR agonists, SARMs, SIRT1 activators, 11beta-HSD1 inhibitors
Incretin/glucagon pathway modulators
Dipeptidyl peptidase-4 inhibitors, glucagon-receptor antagonists
SGLT-2 Inhibitors
Other oral agents
Diacylglycerol acyltransferase and ACC inhibitors, thyroid hormone receptor beta (TRβ) agonists, farnesoid X receptor (FXR) agonists, peroxisome proliferator-activated receptor, niacin derivatives, CCR2 antagonists, ileal bile acid transport (IBAT) inhibitors, PDF4 inhibitors, de novo lipogenesis (DGAT, SCD1 & ACC) inhibitors, cannabinoid 1 receptor modulator

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